PROTAC

Exploration and innovation of Linker features in PROTAC design

Exploration and innovation of Linker features in PROTAC design

Targeted Chimera Proteolysis (PROTAC) technology represents a breakthrough development in the field of drug discovery, utilizing the ubiquitin proteasome system to specifically degrade disease-associated proteins. PROTACs has a two-part function structure, that […]

Four Mechanisms of Action of Molecular Glue

Four Mechanisms of Action of Molecular Glue

Molecular Glue refers to small molecules, typically smaller than PROTACs, often with improved physicochemical properties, designed to stabilize interactions between two proteins. In most cases, this approach is used to enhance […]

New PROTAC Technology

New PROTAC Technology

Protein homeostasis refers to the balance of proteins within cells, involving processes such as protein synthesis, folding, modification, transport, function, and degradation. Proteins in cells participate in nearly all life […]